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KCI 등재
Melanin Biosynthesis Inhibitory Effects of Calycosin-7-O-${\beta}$-D-glucoside Isolated from Astragalus (Astragalus membranaceus)
Kim, Jin-Hee, Lee, Eun-Sook, Lee, Choong-Hwan
DOI http://dx.doi.org/10.1007/s10068-011-0205-4

To discover an active skin depigmentation agent, we isolated a melanin biosynthesis inhibitor from the methanol extract of astragalus (Astragalus membranaceus) using a bioactivity-guided fractionation and identified it as calycosin-7-O-${\beta}$-D-glucoside via spectroscopic analysis. The active compound exhibited tyrosinase inhibitory activity with an $IC_{50}$ value of 68 ${\mu}M$. In addition, calycosin-7-O-${\beta}$-D-glucoside showed a melanin biosynthesis inhibition zone in a culture plate of Streptomyces bikiniensis. Furthermore, 75.78 ${\mu}M$ of calycosin-7-O-${\beta}$-D-glucoside dramatically decreased 50% of the melanin content on Melan-a cells without any apparent cytotoxicity. Theses results indicate that the calycosin-7-O-${\beta}$-D-glucoside isolated from astragalus may be a good candidate for skin-whitening agent.

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