18.97.14.90
18.97.14.90
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케토프로펜 겔제제로부터 약물의 경피흡수
Percutaneous Absorption of Ketoprofen from Gel Preparations
단현광(Hyun - Kwang Tan), 지상철(Sang - Cheol Chi), 전흥원(H . Won Jun)
UCI I410-ECN-0102-2008-510-000804696

In order to reduce the systemic side effects and gastrointestinal irritation of ketoprofen after its oral administration, it was formulated as a 3% ketoprofen gel (ID-GEL) with Pluronic F-127. The pharmacokinetic characteristics of ID-GEL was evaluated following its transdermal application on the dorsal skin of rats at the dose of 9 ㎎/㎏ in reference to those of existing 3% ketoprofen gels. Even though the maximum concentration of 810 ng/㎖ was reached at 6 hrs postdose, the plasma concentration was kept almost constant until 24 hrs postdose, which suggested that ketoprofen was released continuously from the gel during this period. The bioavailability of ID-GEL was two times higher than those of existing 3% ketoprofen gels, based on the calculated area under the plasma concentration-time curves after the percutaneous administration.

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